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氯硝西泮和氯硝西泮区别
更新时间: 2021-04-21 05:59:48  

1、二者均为苯二氮卓类镇静催眠药,在结构上,氯硝西泮比硝西泮多了一个氯。

2、硝西泮的催眠作用更为突出,起效快,引起的睡眠近似生理性,无明显后遗作用,安全范围广,临床上主要用以替代巴比妥类作为催眠药。口服后1~3小时血药浓度达峰值。

3、氯硝西泮特点是抗惊厥作用突出,较硝西泮强5倍,且疗效稳定。此药对呼吸、循环均有抑制作用,且比地西泮强。口服后吸收较慢,2~4小时血药浓度达峰值。临床上对癫痫小发作、婴儿痉挛性及肌阵挛性发作疗效明显,对癫痫持续状态也有效。突然停药可诱发癫痫状态,停药时应逐渐撤停。用于癫痫患者的麻醉前给药,以防止麻醉中及麻醉后的癫痫发作。

关键词: 区别

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